Joan Bosch2012-11-212025-02-172012-11-212012-11-21https://dl.ftveti.edu.et/handle/123456789/3860ÐThe synthesis of 5-(sulfamoylmethyl)indoles bearing a two-carbon chain at C-3 (aminoethyl, acetate, hydroxyethyl, ethyl) either by the Grandberg modi®cation of the Fischer indolization or by intramolecular Heck reaction of suitable o-halotri¯uoroacetanilides is reported. q 2001 Elsevier Science Ltd. All rights reserved.The synthesis of 5-(sulfamoylmethyl)indoles bearing a two-carbon chain at C-3 (aminoethyl, acetate, hydroxyethyl, ethyl) either by the Grandberg modi®cation of the Fischer indolization or by intramolecular Heck reaction of suitable o-halotri¯uoroacetanilides is reported. q 2001 Elsevier Science Ltd. All rights reserved.enSynthesis of 5-(sulfamoylmethyl)indolesArticle