Synthesis of 5-(sulfamoylmethyl)indoles
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Date
2012-11-09
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Abstract
The synthesis of 5-(sulfamoylmethyl)indoles bearing a two-carbon chain at C-3 (aminoethyl, acetate, hydroxyethyl, ethyl) either
by the Grandberg modi®cation of the Fischer indolization or by intramolecular Heck reaction of suitable o-halotri¯uoroacetanilides is
reported. q 2001 Elsevier Science Ltd. All rights reserved
Description
The synthesis of 5-(sulfamoylmethyl)indoles bearing a two-carbon chain at C-3 (aminoethyl, acetate, hydroxyethyl, ethyl) either
by the Grandberg modi®cation of the Fischer indolization or by intramolecular Heck reaction of suitable o-halotri¯uoroacetanilides is
reported. q 2001 Elsevier Science Ltd. All rights reserved.
Keywords
The synthesis of 5-(sulfamoylmethyl)indoles bearing a two-carbon chain at C-3 (aminoethyl, acetate, hydroxyethyl, ethyl) either by the Grandberg modi®cation of the Fischer indolization or by intramolecular Heck reaction of suitable o-halotri¯uoroacetanilides is reported. q 2001 Elsevier Science Ltd. All rights reserved